WebTwo new regioisomers acyclonucleosides bearing 1,2,4-triazole rings as the base moiety were synthesised with aliphatic side chain [(2-acetoxyethoxy)methyl]-bromide under solid-liquid phase transfer catalysis (S.L.P.T.C.) and under silylation method. Biological evaluation of all product revealed they were inactive against various RNA and DNA viruses in cell … WebMay 2, 2014 · The analysis above indicated that the variation of the substituent groups on the 1,2,3-triazole ring had a great effect on the antifungal activity against C. lagenarium. …
Synthesis and Antifungal Activity of Benzamidine Derivatives Carrying 1 …
WebFeb 2, 2024 · In recent years, 1,2,4-triazole derivatives have been extensively studied in many pesticides and pharmaceuticals, and some 1,2,4-triazole drugs have been applied in the clinic. As shown in Scheme 1 a, itraconazole exhibits antimycotic drug activity, ribavirin exhibits antiviral drug activity, and rizatriptan has antimigraine drug activity [7]. WebFeb 27, 2024 · In this atom- and step-economical one-pot process, valuable 1,2,4-triazolo [4,3- a ]pyridines and related heterocyclic compounds could be synthesized efficiently … batterie 92ah agm
Synthesis, antioxidant and anticancer activity of new quinoline-[1, …
WebFeb 19, 2024 · In this review, we have highlighted some recent synthetic approaches for the synthesis of versatile 1,2,4-triazole heterocycles using 3-amino-1,2,4-triazole. 3-Amino-1,2,4-triazole is an effective mono- or bi-nucleophile in controlled multidirectional reactions that lead to the synthesis of a variety of heterocycles with a high number of ... WebA general method for the synthesis of 1,3,5-trisubstituted 1,2,4-triazoles has been developed from reaction of carboxylic acids, ... Environ-Economic Synthesis and Characterization of … WebTwo new regioisomers acyclonucleosides bearing 1,2,4-triazole rings as the base moiety were synthesised with aliphatic side chain [(2-acetoxyethoxy)methyl]-bromide under solid … thijs porck